Reprint

Molecular Methods in Antibiotics Discovery

Edited by
September 2024
224 pages
  • ISBN978-3-7258-2004-7 (Hardback)
  • ISBN978-3-7258-2003-0 (PDF)

This is a Reprint of the Special Issue Molecular Methods in Antibiotics Discovery that was published in

Biology & Life Sciences
Medicine & Pharmacology
Summary

This Special Issue welcomed manuscripts that describe new compounds with antibiotic activity. Eleven papers were published, most of which describe novel compounds, including homopolymers, cyclic imides, antimicrobial peptides, nucleic acids, and derivatives of quinone, benzamidine, thiazole, and pyrazole. Two papers describe novel galenic formulations of titanate or silver nanoparticles, respectively, and one contribution describes repurposed drugs. While most of the contributions to this Special Issue describe compounds with antibacterial activity, two papers describe antimicrobial candidates that have both antibacterial and antifungal properties, and one paper describes compounds with antifungal activity.

Format
  • Hardback
License and Copyright
© 2024 by the authors; CC BY-NC-ND license
Keywords
antibiofilm activity; candidiasis; synergism; synthetic peptides; antifungal drugs; pyrazole; persisters; Staphylococcus aureus; Enterococcus faecalis; resistance; pyrrolidinone; aldol; antibacterial; carbonic anhydrase; sulfonamides; inhibitors; antibiotic resistance; bacteria; 2-aminothiazoles; antifungal; antibacterial; anticancer activity; hydrazone; benzimidazole; sulphanilamide; benzyl alkyl imidazolium ionic liquids; microemulsions; silver nanoparticles; antibacterial; skin bacterial infection treatments; periodontal disease; periodontitis; heterocyclics; antibacterial; benzamidine; bone disorders; bone infections; sodium titanate nanotubes; anti-bacterial; anti-fungal; biomaterial; wound infections; rat model; synthesis; antibacterial agents; quinonic-antibiotics; structure–activity relationships; Craig plot; methicillin-resistant Staphylococcus aureus; Enterococcus faecium; Klebsiella pneumoniae; antibacterial activity; drug discovery; quinone-antibiotics; Free-Wilson; antimicrobial; bactericidal; quaternary ammonium; RAFT polymerization; antisense oligonucleotides; antisense therapies; drug delivery; drug discovery; nucleic acid engineering; ribozymes; riboswitches; n/a

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